ChemicalBook >> CAS DataBase List >>Imidazo[1,2-a]pyridine-5-carbonitrile, 6-amino-3-[3-[(1-aminocyclopentyl)methoxy]-4-cyano-5-(methylthio)phenyl]-
Imidazo[1,2-a]pyridine-5-carbonitrile, 6-amino-3-[3-[(1-aminocyclopentyl)methoxy]-4-cyano-5-(methylthio)phenyl]-
- CAS No.
- 3033846-20-4
- Chemical Name:
- Imidazo[1,2-a]pyridine-5-carbonitrile, 6-amino-3-[3-[(1-aminocyclopentyl)methoxy]-4-cyano-5-(methylthio)phenyl]-
- Synonyms
- SIK-IN-2;Imidazo[1,2-a]pyridine-5-carbonitrile, 6-amino-3-[3-[(1-aminocyclopentyl)methoxy]-4-cyano-5-(methylthio)phenyl]-
- CBNumber:
- CB614214895
- Molecular Formula:
- C22H22N6OS
- Molecular Weight:
- 418.52
- MDL Number:
- MOL File:
- 3033846-20-4.mol
Last updated:2025-04-17 18:22:24
Imidazo[1,2-a]pyridine-5-carbonitrile, 6-amino-3-[3-[(1-aminocyclopentyl)methoxy]-4-cyano-5-(methylthio)phenyl]- Chemical Properties,Uses,Production
Uses
SIK-IN-2 (Compound 45) is an inhibitor for salt-inducible kinase (SIK), which inhibits SKI1, SIK2 and SIK3 with IC50s of 0.1, 0.2 and 0.4 nM, respectively. SIK-IN-2 inhibits the release of TNFa with IC50 of 0.5 nM, stimulates the LPS (HY-D1056) -induced IL-10 release with EC50 of 2 nM in human macrophages[1].
References
[1] Bootsma AN et al., Heterocyclic sik inhibitors. WO2024062360A1.
Imidazo[1,2-a]pyridine-5-carbonitrile, 6-amino-3-[3-[(1-aminocyclopentyl)methoxy]-4-cyano-5-(methylthio)phenyl]- Preparation Products And Raw materials
Raw materials
Preparation Products
Imidazo[1,2-a]pyridine-5-carbonitrile, 6-amino-3-[3-[(1-aminocyclopentyl)methoxy]-4-cyano-5-(methylthio)phenyl]- Suppliers
Global( 1)Suppliers
Supplier | Tel | Country | ProdList | Advantage | |
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TargetMol Chemicals Inc. | 15002134094 | marketing@targetmol.cn | China | 20701 | 58 |
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TargetMol Chemicals Inc. | 58 |
Imidazo[1,2-a]pyridine-5-carbonitrile, 6-amino-3-[3-[(1-aminocyclopentyl)methoxy]-4-cyano-5-(methylthio)phenyl]-
SIK-IN-2
3033846-20-4