
Estrogen receptor modulator 1 NEW
Price | $30 | $58 |
Package | 10mg | 25mg |
Min. Order: | |
Supply Ability: | 10g |
Update Time: | 2025-05-26 |
Product Details
Product Name: Estrogen receptor modulator 1 | CAS No.: 63676-22-2 |
Purity: 98.14% | Supply Ability: 10g |
Release date: 2025/05/26 |
Product Introduction
Bioactivity
Name | Estrogen receptor modulator 1 |
Description | Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.46). |
In vitro | Estrogen receptor modulator 1 (100 nM; 9 days) obviously inhibits the growth of MCF-7:5C cell. It also causes apoptosis in these cells 6 days. Estrogen receptor modulator 1 (100 nM; 10 days) inhibits T47D:A18/PKCα and T47D:A18-TAM1 colony formation [2]. |
In vivo | Estrogen receptor modulator 1 (1.5 mg/animal; p.o.; daily for 2 weeks) induces regression of T47D:A18/PKCα tumors [2]. |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Solubility Information | DMSO : 50 mg/mL (206.36 mM), Sonication is recommended. |
Keywords | tumor | selective | mice | MCF-7:5C | Inhibitor | inhibit | EstrogenReceptor | Estrogen Receptor/ERR | Estrogen receptor modulator-1 | Estrogen receptor modulator1 | Estrogen receptor modulator 1 | Estrogen Receptor | ERR | cells | cancer | breast | athymic |
Inhibitors Related | Kaempferol | Tamoxifen | Estradiol | Estradiol benzoate | ARV-471 | Octinoxate | Genistin | Cholesterol | Estriol | Chrysin | Ethisterone | Estrone |
Related Compound Libraries | Nuclear Receptor Compound Library | Bioactive Compound Library | Membrane Protein-targeted Compound Library | Anti-Ovarian Cancer Compound Library | Endocrinology-Hormone Compound Library | NO PAINS Compound Library | Orally Active Compound Library | Bioactive Compounds Library Max | Anti-Cancer Compound Library | Anti-Cancer Active Compound Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, MA
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