Enalaprilat NEW
| Price | Get Latest Price |
| Package | 1removed |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-05-09 |
Product Details
| Product Name: Enalaprilat | CAS No.: 76420-72-9 |
| Purity: 97.28% | Supply Ability: 10g |
| Release date: 2025/05/09 |
Product Introduction
Bioactivity
| Name | Enalaprilat |
| Description | Enalaprilat (Enalapril acid) is a potent angiotensin-converting enzyme (ACE) inhibitor that enhances arterial and cardiopulmonary pressure reflex control of sympathetic activity in patients with heart failure, and can be used in the study of cardiovascular disease. |
| In vitro | Enalaprilat, the active metabolite of the orally administered drug enalapril, exhibits potent, competitive and long-lasting angiotensin-converting enzyme (ACE) inhibition with an IC50 of 1.94 nM.[1] Enalaprilat (1 nM-10 μM; 24 hours) inhibited IGF-I-induced proliferation of neonatal rat cardiac fibroblasts by 30% in a concentration-dependent manner with an IC50 of 90 nM.[2] |
| In vivo | Enalaprilat (0.01%-2.9% ophthalmic concentration) showed significant IOP-lowering effect in rabbit IOP assay. [3] |
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility Information | DMSO : 80.00 mg/mL (229.63 mM), Sonication is recommended. |
| Keywords | MK 422 | Enalaprilat |
| Inhibitors Related | Olmesartan Medoxomil | Losartan potassium | Tranilast | Enalapril Maleate | Azilsartan Methyl Ester | Sacubitril/Valsartan | Azilsartan | Irbesartan | Losartan | Ramipril | Captopril | Valsartan Methyl Ester |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, USA
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