MIN-101 manufacturers
- Roluperidone
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- $30.00 / 1mg
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2024-11-19
- CAS:359625-79-9
- Min. Order:
- Purity: 97.77%
- Supply Ability: 10g
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| MIN-101 Basic information |
Product Name: | MIN-101 | Synonyms: | MIN-101;CYR-101;Roluperidone (CYR-101);MIN-101; MIN 101; MIN101; CYR-101; CYR 101; CYR101; MT-210; MT 210; MT210;;MT 210;MT210;MT-210;Roluperidone | CAS: | 359625-79-9 | MF: | C22H23FN2O2 | MW: | 366.43 | EINECS: | | Product Categories: | APIS | Mol File: | 359625-79-9.mol |  |
| MIN-101 Chemical Properties |
storage temp. | Store at -20°C | solubility | DMSO:33.33(Max Conc. mg/mL);90.96(Max Conc. mM) | form | A solid | color | White to yellow |
| MIN-101 Usage And Synthesis |
Uses | Roluperidone (CYR-101) is a novel cyclic amide derivative that has high equipotent affinities for 5-HT2A and sigma-2 receptors (Ki of 7.53 nM and 8.19 nM for 5-HT2A and sigma-2, respectively). | IC 50 | 5-HT2A Receptor: 7.53 nM (Ki); Sigma-2 Receptor: 8.19 nM (Ki) | References | [1] Davidson M, et al. Efficacy and Safety of MIN-101: A 12-Week Randomized, Double-Blind, Placebo-Controlled Trial of a New Drug in Development for the Treatment of Negative Symptoms in Schizophrenia. Am J Psychiatry. 2017 Jul 28:appiajp201717010122. DOI:10.1176/appi.ajp.2017.17010122 |
| MIN-101 Preparation Products And Raw materials |
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