Benzonitrile, 2-fluoro-4-[5-(2-methyl-1,3-dioxolan-2-yl)-3-pyridinyl]-
- CAS No.
- 2241573-22-6
- Chemical Name:
- Benzonitrile, 2-fluoro-4-[5-(2-methyl-1,3-dioxolan-2-yl)-3-pyridinyl]-
- Synonyms
- CYP11B2-IN-2;Benzonitrile, 2-fluoro-4-[5-(2-methyl-1,3-dioxolan-2-yl)-3-pyridinyl]-
- CBNumber:
- CB714686222
- Molecular Formula:
- C16H13FN2O2
- Molecular Weight:
- 284.29
- MDL Number:
- MOL File:
- 2241573-22-6.mol
Benzonitrile, 2-fluoro-4-[5-(2-methyl-1,3-dioxolan-2-yl)-3-pyridinyl]- Chemical Properties,Uses,Production
Uses
CYP11B2-IN-2 (Compound 10k) is an inhibitor for enzyme aldosterone synthase CYP11B2 with an IC50 of 0.3 nM. CYP11B2-IN-2 CYP11B-IN-2 is labeled with 18F and can be used as a positron emission tomography (PET) tracer for the diagnosis of primary aldosteronism[1].
IC 50
CYP11B2: 0.3 nM (IC50); CYP11B1: 3.8 nM (IC50)
References
[1] Maier P, et al., Fluorinated aldosterone synthase (CYP11B2)-inhibitors for differential diagnosis between bilateral and unilateral conditions of primary aldosteronism. Bioorg Med Chem Lett. 2023 Nov 15;96:129501. DOI:10.1016/j.bmcl.2023.129501
Benzonitrile, 2-fluoro-4-[5-(2-methyl-1,3-dioxolan-2-yl)-3-pyridinyl]- Preparation Products And Raw materials
Raw materials
Preparation Products
Benzonitrile, 2-fluoro-4-[5-(2-methyl-1,3-dioxolan-2-yl)-3-pyridinyl]- Suppliers
Supplier | Tel | Country | ProdList | Advantage | |
---|---|---|---|---|---|
Shanghai Beckham Medical Technology Co., Ltd | 021-13816613772 13816613772 | huahero21@sina.com | China | 1666 | 55 |
TargetMol Chemicals Inc. | 15002134094 | marketing@targetmol.cn | China | 24803 | 58 |
Supplier | Advantage |
---|---|
Shanghai Beckham Medical Technology Co., Ltd | 55 |
TargetMol Chemicals Inc. | 58 |