| Identification | Back Directory | [Name]
Telapristone | [CAS]
198414-30-1 | [Synonyms]
Telapristone
metabolite of telapristone acetate (CDB-4124)
19-Norpregna-4,9-diene-3,20-dione, 11-[4-(dimethylamino)phenyl]-17-hydroxy-21-methoxy-, (11β)-
(8S,11R,13S,14S,17R)-11-[4-(dimethylamino)phenyl]-17-hydroxy-17-(2-methoxyacetyl)-13-methyl-1,2,6,7,8,11,12,14,15,16-decahydrocyclopenta[a]phenanthren-3-one | [Molecular Formula]
C29H37NO4 | [MDL Number]
MFCD19443748 | [MOL File]
198414-30-1.mol | [Molecular Weight]
463.608 |
| Hazard Information | Back Directory | [Uses]
Telapristone is a Progesterone antagonist. Telapristone can be used in the study of uterine fibroids and endometriosis[1]. | [References]
[1] Morris D, et al. Population pharmacokinetics of telapristone (CDB-4124) and its active monodemethylated metabolite CDB-4453, with a mixture model for total clearance. AAPS J. 2011 Dec;13(4):665-73. DOI:10.1208/s12248-011-9304-7 |
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